SCHEMBL9903994

SCHEMBL9903994

Cn1c(=O)[nH]c(=O)c2c1nc(-c1cn(Cc3cccc(C(F)(F)F)c3)nn1)n2COCC[Si](C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.42
TP53 P04637 2/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
PSEN1 P49768 1/20 0.42
PSEN2 P49810 1/20 0.42
KCNH2 Q12809 1/20 0.42
APH1B Q8WW43 1/20 0.42
NCSTN Q92542 1/20 0.42
APH1A Q96BI3 1/20 0.42
PSENEN Q9NZ42 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
TPH1 P17752 1/20 0.41
TPH2 Q8IWU9 1/20 0.41
KDR P35968 2/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
POLB P06746 2/20 0.39
CXCL8 P10145 1/20 0.39
NOD2 Q9HC29 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904089 0.75 ADORA2B (0.55) PSEN1PSEN2KCNH2APH1BNCSTN
SCHEMBL9904085 0.75 MAOB (0.59) TP53SMN1; SMN2PSEN1PSEN2KCNH2
SCHEMBL21153831 0.69 ADORA2B (0.48) ADORA3ADORA2AADORA2BADORA1
SCHEMBL18833765 0.69 ALDH1A1 (0.48) HPGDALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL16029308 0.69 TRPC1 (0.45) HPGDTP53ALDH1A1SMN1; SMN2KMT2A
SCHEMBL16363925 0.68 MAPK1 (0.46) HPGDTP53ALDH1A1SMN1; SMN2TPH1
SCHEMBL21153830 0.67 ADORA2B (0.51) ADORA3ADORA2AADORA2BADORA1
SCHEMBL9903991 0.67 ADORA2A (0.72) GPR55ADORA3ADORA2AADORA2BADORA1
SCHEMBL23067580 0.67 ADORA2B (0.49) ADORA3ADORA2AADORA2BADORA1
SCHEMBL638535 0.66 MAPT (0.59) HPGDALDH1A1SMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465859-A1 8-Triazolylxanthine derivatives, processes for their production and their use as adenosine receptor antagonists Life & Brain GmbH (DE) 2012-06-20 EP disclosed
WO-2012076974-A1 8-TRIAZOLYLXANTHINE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND THEIR USE AS ADENOSINE RECEPTOR ANTAGONISTS LIFE & BRAIN GMBH (DE) 2012-06-14 WO disclosed