SCHEMBL990901

SCHEMBL990901

Nc1ccc(Nc2ccccc2)cc1C1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.47
GAA P10253 6/20 0.47
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
TDP1 Q9NUW8 4/20 0.47
LMNA P02545 4/20 0.47
KDM4E B2RXH2 3/20 0.47
GFER P55789 2/20 0.47
ALDH1A1 P00352 6/20 0.43
CYP3A4 P08684 4/20 0.43
ALOX12 P18054 3/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
HTT P42858 1/20 0.43
MAPK1 P28482 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
AR P10275 1/20 0.41
HSD17B10 Q99714 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24022743 0.87 TDO2 (0.47) MAPTGAAMEN1KMT2ATDP1
SCHEMBL21779787 0.85 TDO2 (0.46) MAPTGAAMEN1KMT2ATDP1
SCHEMBL6447787 0.75 MAPT (0.41) MAPTGAAMEN1KMT2ATDP1
SCHEMBL21278408 0.75 MAPT (0.48) MAPTGAAMEN1KMT2ATDP1
SCHEMBL1498644 0.75 PDE5A (0.38) MAPTGAAMEN1KMT2ATDP1
SCHEMBL1335958 0.74 NPY5R (0.60) MAPTGAAMEN1KMT2ATDP1
SCHEMBL11199863 0.74 NPY5R (0.60) MAPTGAAMEN1KMT2ATDP1
SCHEMBL3963851 0.74 GAA (0.53) MAPTGAAMEN1KMT2ATDP1
SCHEMBL28690383 0.72 NPY5R (0.57) MAPTGAAMEN1KMT2ATDP1
SCHEMBL5150614 0.72 ALDH1A1 (0.44) MAPTGAAMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 155 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112608402-A Styrene block copolymer and preparation method thereof 北京化工大学 2021-04-06 CN claimed
CN-106661270-A Use of hydroxybenzotriazole derivatives and/or hydroxy indazole derivatives as flame retardants for plastics and flameproof plastic moulded bodies 弗劳恩霍夫应用研究促进协会 2017-05-10 CN claimed
EP-1976821-B1 DIRECT ALKYLATION OF N-ALKYL-N'-PHENYL-P-PHENYLENEDIAMINE CHEMTURA CORP (US) 2011-05-25 EP claimed
EP-1536847-A1 RADIATION STERILIZED MEDICAL DEVICES COMPRISING RADIATION SENSITIVE POLYMERS SCIMED LIFE SYSTEMS, INC. (US) 2005-06-08 EP claimed
WO-2004024204-A1 RADIATION STERILIZED MEDICAL DEVICES COMPRISING RADIATION SENSITIVE POLYMERS SCIMED LIFE SYSTEMS, INC. (US) 2004-03-25 WO claimed
EP-4308638-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING POLYOLEFIN RECYCLATES, STABILIZER COMPOSITION, MASTER BATCH CONCENTRATE, PLASTIC COMPOSITION, MOLDING COMPOUND OR MOLDING, METHOD FOR STABILIZING A POLYOLEFIN RECYCLATE AND USE OF A PLASTIC COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-24 EP disclosed
EP-4308642-A1 STABILIZER COMPOSITION, USE OF THE STABILIZER COMPOSITION, METHOD FOR STABILIZING CONDENSATION POLYMERS AGAINST HYDROLYTIC DEGRADATION, AND HYDROLYSIS-STABILIZED COMPOSITION AND MOLDING OR MOLDED PART CONSISTING THEREOF Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-24 EP disclosed
EP-4305098-A1 USE OF AT LEAST ONE SULFUR-CONTAINING AMINO ACID FOR STABILIZING RECYCLED THERMOPLASTICS, STABILIZED RECYCLED THERMOPLASTIC, STABILIZER COMPOSITION, MASTERBATCH, AND MOLDING COMPOUND OR MOLDED PART Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-17 EP disclosed
EP-4301809-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-10 EP disclosed
WO-2023234394-A1 ASYMMETRIC DIAMINE-CONTAINING AGENT AND RESIN, AND USE THEREOF 住友化学株式会社 2023-12-07 WO disclosed
EP-4237484-A1 USE OF EUGENOL DERIVATIVES AS STABILIZERS, ORGANIC MATERIAL AND EUGENOL DERIVATIVES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-09-06 EP disclosed
EP-4214275-A1 USE OF DIEUGENOL, OLIGOMERS AND/OR POLYMERS OF EUGENOL FOR STABILIZING ORGANIC MATERIALS, STABILIZED PLASTICS COMPOSITION, STABILIZER COMPOSITION AND METHOD FOR STABILIZING ORGANIC MATERIALS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-07-26 EP disclosed
EP-1149122-A1 TACK FREE SURFACE CURES OF POLYMERS BY ORGANIC PEROXIDES IN THE PRESENCE OF AIR Atofina Chemicals, Inc. (US) 2001-10-31 EP disclosed
WO-2001058987-A2 HYPERBRANCHED AMPHIPHILIC POLYMERIC ADDITIVES AND POLYMER COMPOSITIONS WITH INCREASED SURFACE ENERGY CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2001-08-16 WO disclosed
WO-2001034680-A1 TACK FREE SURFACE CURES OF POLYMERS BY ORGANIC PEROXIDES IN THE PRESENCE OF AIR ATOFINA CHEMICALS, INC. (US) 2001-05-17 WO disclosed
EP-1036081-A1 HETEROCYCLYL LIGAND CONTAINING RUTHENIUM AND OSMIUM CATALYSTS Ciba SC Holding AG (CH) 2000-09-20 EP disclosed
EP-0994855-A1 LIGHT-STABILIZING SYNERGIC MIXTURES FOR ORGANIC POLYMERS Great Lakes Chemical (Europe) GmbH (CH) 2000-04-26 EP disclosed
WO-1999048997-A1 STABILISATION OF ORGANIC MATERIALS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-09-30 WO disclosed
WO-1999029701-A1 HETEROCYCLYL LIGAND CONTAINING RUTHENIUM AND OSMIUM CATALYSTS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-06-17 WO disclosed
WO-1999002495-A1 LIGHT-STABILIZING SYNERGIC MIXTURES FOR ORGANIC POLYMERS GREAT LAKES CHEMICAL (EUROPE) GMBH (CH) 1999-01-21 WO disclosed