SCHEMBL9911342

SCHEMBL9911342

Cc1ccc(CNC(C)C)cc1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.46
PTGS1 P23219 1/20 0.46
CACNA1C Q13936 1/20 0.46
ERCC1 P07992 2/20 0.44
ERCC4 Q92889 2/20 0.44
MEN1 O00255 4/20 0.40
CYP3A4 P08684 4/20 0.40
KMT2A Q03164 4/20 0.40
ALOX15 P16050 3/20 0.40
ALOX12 P18054 3/20 0.40
ESR1 P03372 3/20 0.40
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
MAPK1 P28482 3/20 0.40
HIF1A Q16665 3/20 0.40
HSD17B10 Q99714 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2C19 P33261 3/20 0.40
TP53 P04637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9911520 0.85 ERCC1 (0.59) TRPA1ERCC1ERCC4MEN1CYP3A4
SCHEMBL12312617 0.82 SLC2A1 (0.42) MEN1CYP3A4KMT2AALDH1A1CYP1A2
SCHEMBL15981393 0.79 ERCC1 (0.49) TRPA1ERCC1ERCC4MEN1CYP3A4
SCHEMBL17576040 0.79 ESR1 (0.47) TRPA1PTGS1CACNA1CERCC1ERCC4
SCHEMBL28285719 0.78 GABRA1 (0.50) TRPA1ERCC1ERCC4MEN1CYP3A4
Hydrochloric Acid SCHEMBL1000376 0.76 SLC2A1 (0.41) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL18251691 0.76 ERCC1 (0.77) ERCC1ERCC4MEN1CYP3A4KMT2A
SCHEMBL13881303 0.75 MEN1 (0.51) MEN1KMT2AALOX15KDM4EALDH1A1
SCHEMBL28259627 0.75 ERCC1 (0.39) TRPA1ERCC1ERCC4MEN1CYP3A4
SCHEMBL3271284 0.75 SIGMAR1 (0.48) ALOX15ALDH1A1MAPK1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed