SCHEMBL9911486

SCHEMBL9911486

CC(C)NC(=O)CNc1cc[n+]([O-])cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
PKM P14618 2/20 0.40
ALDH1A1 P00352 7/20 0.38
MAPT P10636 3/20 0.38
NLRP1 Q9C000 1/20 0.38
KDM1A O60341 1/20 0.38
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36
HPGD P15428 2/20 0.35
LMNA P02545 3/20 0.34
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
FFAR1 O14842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24137901 0.80 LMNA (0.51) KMT2AMEN1PKMALDH1A1MAPT
SCHEMBL9911482 0.77 GAA (0.46) KMT2AALDH1A1MAPTNLRP1GAA
SCHEMBL6510629 0.74 ALDH1A1 (0.59) KMT2AMEN1PKMALDH1A1MAPT
SCHEMBL9911453 0.70 KMT2A (0.53) KMT2AMEN1ALDH1A1MAPTCA1
SCHEMBL19634841 0.70 NOTUM (0.53) KMT2AMEN1PKMALDH1A1LMNA
SCHEMBL22544884 0.68 KMT2A (0.50) KMT2AMEN1ALDH1A1LMNAGAA
SCHEMBL6623667 0.67 PKM (0.49) KMT2AMEN1PKMALDH1A1MAPT
SCHEMBL13867734 0.67 TDP1 (0.52) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL9835275 0.66 MEN1 (0.45) KMT2AMEN1ALDH1A1KDM1ACA12
SCHEMBL9329532 0.65 PKM (0.47) KMT2AMEN1PKMALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-7300948-B2 Alkynyl compounds as non nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-11-27 US disclosed