SCHEMBL9912183

SCHEMBL9912183

CS(=O)(=O)Nc1ccccc1-c1cc(NCCc2ccc(O)cc2)nc(O)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
MTOR P42345 1/20 0.51
RAB9A P51151 1/20 0.51
SIRT2 Q8IXJ6 1/20 0.51
PTGDR Q13258 4/20 0.46
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PGAM1 P18669 1/20 0.40
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
ADRA1A P35348 2/20 0.39
CXCR2 P25025 1/20 0.39
MCL1 Q07820 1/20 0.38
JAK2 O60674 2/20 0.37
JAK1 P23458 2/20 0.37
TYK2 P29597 2/20 0.37
JAK3 P52333 2/20 0.37
CDK1 P06493 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4496591 0.78 PTGDR (0.70) PTGDR
SCHEMBL9912239 0.72 PTGDR (0.63) NPC1MTORRAB9ASIRT2PTGDR
SCHEMBL13895137 0.71 PTGDR (0.64) PTGDRALDH1A1SMN1; SMN2KDM4EF13A1
SCHEMBL13895143 0.71 ALDH1A1 (0.55) RAB9APTGDRALDH1A1SMN1; SMN2KDM4E
SCHEMBL9912208 0.71 PTGDR (0.57) PTGDRALDH1A1SMN1; SMN2KDM4E
SCHEMBL9912204 0.70 PTGDR (0.56) PTGDRALDH1A1SMN1; SMN2
SCHEMBL13895136 0.70 PTGDR (0.61) NPC1MTORRAB9ASIRT2PTGDR
SCHEMBL13895060 0.70 PTGDR (0.61) PTGDRALDH1A1SMN1; SMN2KDM4E
SCHEMBL9912237 0.70 PTGDR (0.52) PTGDRALDH1A1SMN1; SMN2
SCHEMBL13894988 0.70 CNR2 (0.44) NPC1MTORRAB9ASIRT2PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193183-B2 2,6-substituted-4-monosubstitutedamino-pyrimidine as prostaglandin D2 receptor antagonists AVENTIS PHARMACEUTICALS INC. (US) 2012-06-05 US disclosed
US-7517889-B2 2,6-substituted-4-monosubstitutedamino-pyrimidine as prostaglandin D2 receptor antagonists AVENTIS PHARMACEUTICALS, INC. (US) 2009-04-14 US disclosed