SCHEMBL9921630

SCHEMBL9921630

CCC[C@@H](CNC(=O)Nc1ccccc1)N(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.51
ALDH1A1 P00352 2/20 0.51
HTT P42858 1/20 0.51
KDM4E B2RXH2 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NOX1 Q9Y5S8 1/20 0.47
OPRM1 P35372 5/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46
OPRD1 P41143 4/20 0.45
OPRK1 P41145 4/20 0.45
TP53 P04637 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 1/20 0.44
EPHX2 P34913 1/20 0.44
CDK9 P50750 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11586099 0.75 EPHX1 (0.55) EPHX1ALDH1A1HTTKDM4EL3MBTL1
SCHEMBL10596294 0.75 LMNA (0.61) EPHX1ALDH1A1HTTKDM4ENPC1
SCHEMBL11814215 0.74 ALDH1A1 (0.58) EPHX1ALDH1A1HTTKDM4EL3MBTL1
SCHEMBL7749716 0.73 EPHX1 (0.55) EPHX1ALDH1A1HTTKDM4ENPC1
SCHEMBL17596717 0.73 EPHX1 (0.55) EPHX1ALDH1A1HTTKDM4ENPC1
SCHEMBL17596716 0.73 EPHX1 (0.55) EPHX1ALDH1A1HTTKDM4ENPC1
SCHEMBL28914992 0.73 OPRM1 (0.62) NPC1RAB9AOPRM1OPRD1OPRK1
SCHEMBL2451040 0.73 EPHX1 (0.75) EPHX1ALDH1A1HTTKDM4EL3MBTL1
SCHEMBL8282413 0.73 EPHX1 (0.50) EPHX1ALDH1A1HTTKDM4ENPC1
SCHEMBL7610023 0.73 MEN1 (0.51) ALDH1A1KDM4EL3MBTL1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010185-B1 DIHYDROTHIENOPYRIMIDINE FOR TREATING INFLAMMATORY DISORDERS BOEHRINGER INGELHEIM INT (DE) 2012-06-13 EP disclosed