SCHEMBL9924103

SCHEMBL9924103

CC(C)(C)C(c1ccc(C#N)cc1)c1ccc(OCc2ncccn2)cn1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.40
FFAR1 O14842 1/20 0.39
MAOB P27338 1/20 0.38
CYP4F2 P78329 2/20 0.38
CYP4A11 Q02928 2/20 0.38
NR1H4 Q96RI1 1/20 0.33
S1PR1 P21453 2/20 0.33
S1PR3 Q99500 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2995380 0.89 CYP19A1 (0.45) CYP19A1FFAR1MAOBNR1H4
SCHEMBL9924105 0.88 FFAR1 (0.46) CYP19A1FFAR1MAOBCYP4F2CYP4A11
SCHEMBL9924104 0.85 APP (0.35)
SCHEMBL9924102 0.83 ACACB (0.40) CYP19A1FFAR1MAOBCYP4F2CYP4A11
SCHEMBL2795215 0.82 CYP11B1 (0.43) CYP19A1FFAR1MAOB
SCHEMBL14923018 0.77 CYP19A1 (0.35) CYP19A1MAOBCYP4F2CYP4A11
SCHEMBL2246114 0.76 FFAR1 (0.49) CYP19A1FFAR1MAOB
SCHEMBL9924098 0.74 ALOX5AP (0.48) CYP19A1FFAR1MAOBCYP4F2CYP4A11
SCHEMBL3000768 0.73 MAOB (0.43) CYP19A1FFAR1MAOBNR1H4
SCHEMBL3626112 0.73 MAOB (0.49) CYP19A1FFAR1MAOBCYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8426413-B2 Diaryl substituted alkanes MERCK SHARP & DOHME CORP. (US) 2013-04-23 US disclosed
US-8426413-B2 Diaryl substituted alkanes MERCK SHARP & DOHME CORP. (US) 2013-04-23 US disclosed
US-20120149674-A1 Diaryl Substituted Alkanes MERCK SHARPE & DOHME CORP. (US) 2012-06-14 US disclosed
US-20120149674-A1 Diaryl Substituted Alkanes MERCK SHARPE & DOHME CORP. (US) 2012-06-14 US disclosed
US-8124628-B2 Diaryl substituted alkanes MERCK SHARP & DOHME CORP. (US) 2012-02-28 US disclosed
US-8124628-B2 Diaryl substituted alkanes MERCK SHARP & DOHME CORP. (US) 2012-02-28 US disclosed
US-20090258851-A1 DIARYL SUBSTITUTED ALKANES MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
US-20090258851-A1 DIARYL SUBSTITUTED ALKANES MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
WO-2007120574-A2 DIARYL SUBSTITUTED ALKANES MERCK & CO., INC. (US) 2007-10-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149674-A1 Diaryl Substituted Alkanes ALOX5, ALOX15, LTB4R2 CYP19A1 792/4885FFAR1 161/4885MAOB 813/4885
US-20090258851-A1 DIARYL SUBSTITUTED ALKANES ALOX5, ALOX15, LTB4R2 CYP19A1 792/4885FFAR1 161/4885MAOB 813/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.