SCHEMBL9925473

SCHEMBL9925473

Cc1ccc(-c2ccnc3c(C)cc(C(=O)N=O)cc23)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.39
KDM1A O60341 4/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
PTGDR2 Q9Y5Y4 4/20 0.38
CYP2C9 P11712 1/20 0.38
PTGS1 P23219 1/20 0.38
SLC6A4 P31645 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGS2 P35354 1/20 0.38
MAPK14 Q16539 3/20 0.37
GRM2 Q14416 2/20 0.37
CTSA P10619 1/20 0.35
JAK2 O60674 1/20 0.34
DYRK1A Q13627 1/20 0.33
ROCK2 O75116 1/20 0.33
MAP4K4 O95819 1/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9907850 0.88 HTR5A (0.44) HDAC1KDM1AHDAC6HDAC2HDAC11
SCHEMBL9907492 0.87 PTGDR2 (0.42) HDAC1KDM1AHDAC6HDAC2HDAC11
SCHEMBL9907489 0.84 MAPK14 (0.42) HDAC1KDM1AHDAC6HDAC2HDAC11
SCHEMBL9907826 0.79 HTR5A (0.51) MAPK14
SCHEMBL9907849 0.77 HTR5A (0.45) GRM2
SCHEMBL9907490 0.75 KMO (0.48) PTGDR2PTGS1MAPK14GRM2
SCHEMBL9907841 0.75 HTR5A (0.48) PTGDR2CYP2C9PTGS1SLC6A4CYP2C19
SCHEMBL9925360 0.75 MAPK14 (0.41) MAPK14
SCHEMBL9907431 0.74 MAPK14 (0.51) MAPK14
SCHEMBL9907852 0.74 HTR5A (0.41) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463276-A1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2012-06-13 EP disclosed