SCHEMBL9928559

SCHEMBL9928559

Cc1ccccc1-c1cn(-c2nc3c([nH]2)c(=O)n(C)c(=O)n3C)nn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
TDP1 Q9NUW8 1/20 0.49
ADORA2B P29275 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP1A2 P05177 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA1 P30542 1/20 0.47
BLM P54132 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 1/20 0.47
DCTPP1 Q9H773 1/20 0.47
USP2 O75604 1/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
GFER P55789 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904113 0.87 KDM4E (0.49) KDM4EALDH1A1HPGDTDP1ADORA2B
SCHEMBL9904115 0.86 KDM4E (0.47) KDM4EALDH1A1HPGDTDP1ADORA2B
SCHEMBL9928563 0.83 GAA (0.56) KDM4EALDH1A1HPGDTDP1ADORA2B
SCHEMBL9943454 0.81 ALDH1A1 (0.64) KDM4EALDH1A1ADORA2BHSD17B10CYP1A2
SCHEMBL9904126 0.80 DCTPP1 (0.56) KDM4EALDH1A1HPGDADORA2BHSD17B10
SCHEMBL9904312 0.79 ADORA2B (0.48) KDM4EALDH1A1ADORA2BHSD17B10CYP1A2
SCHEMBL9904008 0.79 MAPT (0.57) KDM4EALDH1A1HPGDTDP1ADORA2B
SCHEMBL9928556 0.78 ADORA2B (0.61) KDM4EALDH1A1ADORA2BCYP1A2ADORA2A
SCHEMBL9928558 0.78 ADORA2A (0.43) KDM4EADORA2BHSD17B10CYP1A2ADORA3
SCHEMBL9904107 0.78 ADORA2B (0.46) KDM4EALDH1A1HPGDADORA2BHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076974-A1 8-TRIAZOLYLXANTHINE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND THEIR USE AS ADENOSINE RECEPTOR ANTAGONISTS LIFE & BRAIN GMBH (DE) 2012-06-14 WO disclosed