SCHEMBL9929088

SCHEMBL9929088

COc1ccc(C(=O)c2cccc(C(F)(F)F)c2)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.65
CYP3A4 P08684 2/20 0.65
CYP2C9 P11712 1/20 0.65
TSHR P16473 1/20 0.65
CYP2C19 P33261 1/20 0.65
SRD5A2 P31213 1/20 0.61
NQO2 P16083 1/20 0.60
ALDH1A1 P00352 2/20 0.56
GAA P10253 1/20 0.56
CES2 O00748 1/20 0.54
MAPT P10636 2/20 0.53
POLB P06746 1/20 0.53
MAOB P27338 1/20 0.52
KMT2A Q03164 2/20 0.52
NPSR1 Q6W5P4 1/20 0.51
MEN1 O00255 1/20 0.51
ADORA1 P30542 1/20 0.51
HSD17B10 Q99714 1/20 0.51
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11506232 0.89 SRD5A2 (0.58) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL1962189 0.88 CYP1A2 (0.69) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL15988788 0.87 CTNNB1 (0.67) TSHRNQO2ALDH1A1CES2MAPT
SCHEMBL3962287 0.86 CYP1A2 (0.71) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL8937269 0.84 NQO2 (0.56) SRD5A2NQO2CES2MAPTPOLB
SCHEMBL8937272 0.84 NQO2 (0.56) SRD5A2NQO2CES2MAPTPOLB
SCHEMBL8937264 0.84 NQO2 (0.56) SRD5A2NQO2CES2MAPTPOLB
SCHEMBL7485522 0.84 SRD5A2 (0.68) CYP1A2CYP3A4SRD5A2ALDH1A1GAA
SCHEMBL1237189 0.82 SRD5A2 (0.79) CYP1A2CYP3A4SRD5A2ALDH1A1CES2
SCHEMBL4710822 0.82 MEN1 (0.54) CYP1A2CYP3A4SRD5A2NQO2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651912-B1 PHOTOCHROMIC COMPOUNDS AND COMPOSITIONS TRANSITIONS OPTICAL INC (US) 2018-10-03 EP disclosed
US-9034219-B2 Photochromic compounds and compositions TRANSITIONS OPTICAL, INC. (US) 2015-05-19 US disclosed
US-20120156521-A1 PHOTOCHROMIC COMPOUNDS AND COMPOSITIONS TRANSITIONS OPTICAL, INC. (US) 2012-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120156521-A1 PHOTOCHROMIC COMPOUNDS AND COMPOSITIONS CRY2, CRY1, PPOX CYP1A2 139/4885CYP3A4 595/4885CYP2C9 167/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.