SCHEMBL9938408

SCHEMBL9938408

COC(=O)C(=CN(C)C)C(=O)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.48
RECQL P46063 1/20 0.46
PTPN2 P17706 1/20 0.45
PTPN1 P18031 1/20 0.45
PTPN6 P29350 1/20 0.45
EPHX1 P07099 1/20 0.43
STS P08842 8/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ABL1 P00519 1/20 0.40
RIN1 Q13671 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20428017 0.87 HPGD (0.45) HPGDRECQLPTPN2PTPN1PTPN6
SCHEMBL9971129 0.81 HPGD (0.46) HPGDRECQLPTPN2PTPN1PTPN6
SCHEMBL1015830 0.79 MAPT (0.36) RECQLKMT2AKDM4EMAPT
SCHEMBL31587724 0.79 MAPT (0.36) RECQLKMT2AKDM4EMAPT
SCHEMBL1015828 0.79 MAPT (0.36) RECQLKMT2AKDM4EMAPT
SCHEMBL2515709 0.78
SCHEMBL2515711 0.78
SCHEMBL1014889 0.76 MAPT (0.35) MAPT
SCHEMBL1016151 0.76 CES2 (0.39) ALDH1A1MAPTRAB9A
SCHEMBL17109784 0.76 HPGD (0.55) HPGDRECQLPTPN2PTPN1PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082947-A1 COMPOUNDS AND COMPOSITIONS AS TGR5 AGONISTS IRM LLC (BM) 2012-06-21 WO disclosed