SCHEMBL9938491

SCHEMBL9938491

COc1cc(C(=O)O)cc(-c2ccc(C#N)cc2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.64
PTPN11 Q06124 1/20 0.47
MMP2 P08253 1/20 0.47
PLAU P00749 1/20 0.46
MAPT P10636 2/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
CNR1 P21554 1/20 0.45
CASP1 P29466 1/20 0.45
CNR2 P34972 1/20 0.45
CASP7 P55210 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
THRB P10828 1/20 0.45
PTGER4 P35408 1/20 0.45
NR3C2 P08235 1/20 0.45
XDH P47989 1/20 0.45
MAP4K4 O95819 1/20 0.45
ABL1 P00519 1/20 0.45
ABCB1 P08183 1/20 0.45
BCR P11274 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2516130 0.85 DHODH (0.53) RXRAMMP2XDHMAP4K4EGLN2
SCHEMBL14150399 0.82 RXRA (0.69) RXRACYP3A4SMN1; SMN2HSD17B1HSD17B2
SCHEMBL30420728 0.82 RXRA (0.69) RXRACYP3A4SMN1; SMN2HSD17B1HSD17B2
SCHEMBL16195103 0.81 DHODH (0.56) RXRASMN1; SMN2PTGER4XDHMAP4K4
SCHEMBL2958179 0.81 RXRA (0.68) RXRAABL1ABCB1BCRHSD17B1
SCHEMBL2558136 0.81 RXRA (0.73) RXRAMAPTSMN1; SMN2ABL1ABCB1
SCHEMBL933732 0.80 RXRA (0.51) RXRA
SCHEMBL2561821 0.79 RXRA (0.64) RXRAXDHABL1ABCB1BCR
SCHEMBL2035502 0.79 RXRA (1.00) RXRAMAP4K4ABL1ABCB1BCR
SCHEMBL7157751 0.79 RXRA (0.68) RXRASMN1; SMN2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083145-A1 GLUCOSAMINE DERIVATIVES GLAXO WELLCOME MANUFACTURING PTE LTD (SG) 2012-06-21 WO disclosed
WO-2012083145-A1 GLUCOSAMINE DERIVATIVES GLAXO WELLCOME MANUFACTURING PTE LTD (SG) 2012-06-21 WO disclosed