SCHEMBL9939773

SCHEMBL9939773

NC1(C(=O)NCc2ccc(Cl)c(Nc3nc4cc(N5CCCC5)ccc4[nH]3)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 6/20 0.42
ENPP2 Q13822 4/20 0.37
CNR1 P21554 2/20 0.37
AKT1 P31749 3/20 0.37
ROCK2 O75116 1/20 0.37
CYP2C9 P11712 1/20 0.37
KCNH2 Q12809 1/20 0.37
AKT3 Q9Y243 1/20 0.37
TRPV1 Q8NER1 4/20 0.36
PTGES O14684 1/20 0.36
WDR5 P61964 1/20 0.35
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9939775 0.89 DRD2 (0.40) ENPP2CNR1TRPV1PTGESWDR5
SCHEMBL14238211 0.88 CNR1 (0.36) ENPP2CNR1TRPV1PTGESWDR5
SCHEMBL9939974 0.85 PTGES (0.43) ENPP2CNR1PTGES
SCHEMBL9941944 0.84 SMO (0.44) ENPP2CNR1PTGESMEN1LMNA
SCHEMBL9939834 0.83 PTGES (0.38) ENPP2CNR1TRPV1PTGESWDR5
SCHEMBL9939776 0.83 PTGES (0.38) ENPP2CNR1TRPV1PTGESWDR5
SCHEMBL9939831 0.82 PTGES (0.41) ENPP2CNR1PTGES
SCHEMBL9899450 0.82 MAP2K7 (0.41) CNR1KCNH2HTTSMN1; SMN2
SCHEMBL9939772 0.82 PPARD (0.39) ENPP2CNR1PTGESWDR5
SCHEMBL9939824 0.82 POLB (0.45) ROCK2WDR5MEN1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076672-A1 2 -AMINOBENZ IMIDAZOLE DERIVATIVES USEFUL IN THE TREATMENT OF INFLAMMATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed