SCHEMBL9940508

SCHEMBL9940508

CN(C(=O)CCc1ccccn1)c1cscn1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 5/20 0.39
TDP1 Q9NUW8 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HSD11B1 P28845 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26319974 0.77 CYP1A2 (0.51) HIF1ANPC1POLBRAB9ASMN1; SMN2
SCHEMBL3160952 0.73 KDM4E (0.40) KDM4EALDH1A1
SCHEMBL895535 0.72 HIF1A (0.49) HIF1ANPC1POLBRAB9ASMN1; SMN2
SCHEMBL2722250 0.69 ALDH1A1 (0.57) SMN1; SMN2CYP1A2CYP2C19TDP1ALDH1A1
SCHEMBL5493166 0.69 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2CYP1A2CYP2C19
SCHEMBL403460 0.69 CYP1A2 (0.56) SMN1; SMN2CYP1A2CYP2C19TDP1ALDH1A1
SCHEMBL3161028 0.69 KDM4E (0.41) NPC1POLBRAB9ASMN1; SMN2CYP1A2
SCHEMBL27763463 0.68 MAPK1 (0.38) NPC1RAB9ASMN1; SMN2CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL3001066 0.68 SMN1; SMN2 (0.54) NPC1RAB9ASMN1; SMN2CYP1A2CYP2C19
SCHEMBL29499090 0.67 SMN1; SMN2 (0.62) SMN1; SMN2CYP1A2CYP2C19TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651930-A1 BIARYLAMIDE INHIBITORS OF LEUKOTRIENE PRODUCTION Boehringer Ingelheim International GmbH (DE) 2013-10-23 EP disclosed
WO-2012082817-A1 BIARYLAMIDE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-21 WO disclosed