SCHEMBL99412

SCHEMBL99412

O=C(O)Nc1cc(CCCC(=O)Nc2ccc3cc(CO)ccc3c2)ccc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.47
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
POLB P06746 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
LMNA P02545 2/20 0.45
CYP1A2 P05177 2/20 0.44
HDAC1 Q13547 4/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
MEN1 O00255 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99215 0.94 AKR1C3 (0.49) HCAR2LMNACYP1A2HDAC1MEN1
SCHEMBL101223 0.90 HDAC1 (0.51) NPC1RAB9APOLBSMN1; SMN2HDAC1
SCHEMBL101623 0.87 HDAC2 (0.48) HCAR2SMN1; SMN2HDAC1HDAC2HDAC8
SCHEMBL101227 0.84 NPC1 (0.45) HCAR2NPC1RAB9APOLBSMN1; SMN2
SCHEMBL98208 0.84 HCAR2 (0.41) HCAR2NPC1RAB9APOLBSMN1; SMN2
SCHEMBL98704 0.83 AKR1C3 (0.51) HCAR2NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL100635 0.83 MEN1 (0.48) HCAR2NPC1RAB9APOLBLMNA
SCHEMBL102437 0.83 RORC (0.48) NPC1RAB9APOLBSMN1; SMN2LMNA
SCHEMBL15822177 0.82 HDAC1 (0.47) HCAR2NPC1RAB9APOLBSMN1; SMN2
SCHEMBL100918 0.82 AKR1C3 (0.46) HCAR2NPC1RAB9ASMN1; SMN2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed