SCHEMBL9942722

SCHEMBL9942722

COc1ccc(C#CC(O)c2ccc(OC)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.53
ACACB O00763 2/20 0.50
AOC3 Q16853 2/20 0.45
KCNH2 Q12809 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP19A1 P11511 1/20 0.40
MCHR1 Q99705 1/20 0.40
FFAR1 O14842 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3924311 0.92 APP (0.46) APPACACBAOC3ALDH1A1MAPK1
SCHEMBL23572596 0.91 APP (0.49) APPACACBKCNH2ALDH1A1
SCHEMBL2685285 0.91 APP (0.49) APPACACBKCNH2ALDH1A1
SCHEMBL2683955 0.91 KMT2A (0.47) APPACACBALDH1A1TSHRMAPK1
SCHEMBL22122696 0.91 KMT2A (0.47) APPACACBALDH1A1TSHRMAPK1
SCHEMBL1818040 0.88 FAAH (0.48) APPACACBMAPK1MCHR1
SCHEMBL1819985 0.88 MCHR1 (0.48) APPACACBAOC3ALDH1A1TSHR
SCHEMBL5194250 0.87 CA12 (0.46) APPACACBAOC3CA12CA1
SCHEMBL7053252 0.84 IGF1R (0.45) ALDH1A1MAPK1L3MBTL1
SCHEMBL7734103 0.83 MAPT (0.46) ALDH1A1MAPK1L3MBTL1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2652552-A1 PHOTOCHROMIC COMPOUNDS AND COMPOSITIONS Transitions Optical, Inc. (US) 2013-10-23 EP disclosed
WO-2013032608-A1 INDENO-FUSED RING COMPOUNDS TRANSITIONS OPTICAL, INC. (US) 2013-03-07 WO disclosed
WO-2012082299-A1 PHOTOCHROMIC COMPOUNDS AND COMPOSITIONS TRANSITIONS OPTICAL, INC. (US) 2012-06-21 WO disclosed