SCHEMBL9943304

SCHEMBL9943304

O=c1[nH]c2ccccc2n1C1CCN(CC2COc3ccccc3O2)CC1

nearest known ligand 0.79

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.61
HTR1A P08908 1/20 0.61
HTR2A P28223 1/20 0.61
HTR2C P28335 1/20 0.61
HTR2B P41595 1/20 0.61
OPRM1 P35372 2/20 0.61
OPRK1 P41145 2/20 0.61
OPRL1 P41146 2/20 0.61
CHRM1 P11229 1/20 0.57
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11096032 0.99 DRD2 (0.61) DRD2HTR1AHTR2AHTR2CHTR2B
SCHEMBL11096050 0.90 DRD2 (0.62) DRD2HTR1AHTR2AHTR2CHTR2B
SCHEMBL11664292 0.90 CHRM1 (0.60) DRD2OPRM1OPRK1OPRL1CHRM1
SCHEMBL11101398 0.89 DRD2 (0.62) DRD2HTR1AHTR2AHTR2CHTR2B
SCHEMBL11095945 0.89 DRD2 (0.62) DRD2HTR1AHTR2AHTR2CHTR2B
SCHEMBL11098294 0.89 OPRM1 (0.62) DRD2HTR1AHTR2AHTR2CHTR2B
SCHEMBL11097105 0.89 OPRM1 (0.66) DRD2HTR1AHTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL11257252 0.89 CHRM1 (0.59) DRD2OPRM1OPRK1OPRL1CHRM1
SCHEMBL11024037 0.88 OPRM1 (0.58) DRD2HTR1AHTR2AHTR2CHTR2B
SCHEMBL11101393 0.88 DRD2 (0.59) DRD2HTR1AHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed
EP-0068261-A1 N-oxacyclyl-alkylpiperidine derivatives, their preparation, pharmaceutical preparations containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1983-01-05 EP disclosed