SCHEMBL11096050

SCHEMBL11096050

Cc1cc2c(cc1C)OC(CN1CCC(n3c(=O)[nH]c4ccccc43)CC1)CO2

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.62
HTR2C P28335 2/20 0.62
HTR1A P08908 1/20 0.62
HTR2A P28223 1/20 0.62
HTR2B P41595 1/20 0.62
OPRM1 P35372 5/20 0.57
OPRK1 P41145 3/20 0.57
OPRL1 P41146 3/20 0.57
CHRM2 P08172 2/20 0.56
CHRM5 P08912 2/20 0.56
CHRM1 P11229 2/20 0.56
ADRA1D P25100 2/20 0.56
ADRA1A P35348 2/20 0.56
ADRA1B P35368 2/20 0.56
CHRM4 P08173 1/20 0.56
CHRM3 P20309 1/20 0.56
HTR7 P34969 1/20 0.56
DRD3 P35462 1/20 0.56
OPRD1 P41143 1/20 0.56
CYP2D6 P10635 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11101398 0.92 DRD2 (0.62) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL11095945 0.92 DRD2 (0.62) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL11097105 0.91 OPRM1 (0.66) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL9943304 0.90 DRD2 (0.61) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL11024847 0.89 OPRM1 (0.54) DRD2HTR2CHTR1AHTR2AHTR2B
Hydrochloric Acid SCHEMBL11096032 0.89 DRD2 (0.61) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL11024716 0.88 CHRM1 (0.58) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL11098294 0.88 OPRM1 (0.62) DRD2HTR2CHTR1AHTR2AHTR2B
SCHEMBL11027738 0.88 HTR1A (0.60) DRD2HTR1AHTR2AOPRM1CHRM1
SCHEMBL11103249 0.87 DRD2 (0.59) DRD2HTR2CHTR1AHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4470989-A Neuroleptic n-oxacyclyl-alkylpiperidine derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1984-09-11 US disclosed
EP-0068261-A1 N-oxacyclyl-alkylpiperidine derivatives, their preparation, pharmaceutical preparations containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1983-01-05 EP disclosed