SCHEMBL9945003

SCHEMBL9945003

CNc1cc(Cl)c(C(=O)N[C@H]2CC[C@@H](C)CC2)cc1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
HPGD P15428 3/20 0.47
RAB9A P51151 6/20 0.43
NPC1 O15118 5/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
MITF O75030 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
USP7 Q93009 1/20 0.39
USP47 Q96K76 1/20 0.39
P2RX7 Q99572 1/20 0.39
HCAR3 P49019 1/20 0.38
CDC25B P30305 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9944747 1.00 ALDH1A1 (0.53) ALDH1A1HPGDRAB9ANPC1TAS1R3
SCHEMBL1728088 0.91 NPC1 (0.52) ALDH1A1HPGDRAB9ANPC1SMN1; SMN2
SCHEMBL9944880 0.88 ALDH1A1 (0.50) ALDH1A1HPGDRAB9ANPC1TAS1R3
SCHEMBL9897509 0.87 ALDH1A1 (0.49) ALDH1A1HPGDRAB9ANPC1SMN1; SMN2
SCHEMBL9897513 0.87 ALDH1A1 (0.49) ALDH1A1HPGDRAB9ANPC1SMN1; SMN2
SCHEMBL9944736 0.86 ALDH1A1 (0.47) ALDH1A1HPGDRAB9ANPC1TAS1R3
SCHEMBL12494909 0.84 ALDH1A1 (0.59) ALDH1A1HPGDRAB9ANPC1SMN1; SMN2
SCHEMBL9945024 0.84 ALDH1A1 (0.47) ALDH1A1HPGDRAB9ANPC1TAS1R3
SCHEMBL9945014 0.84 ALDH1A1 (0.47) ALDH1A1HPGDRAB9ANPC1TAS1R3
SCHEMBL9945010 0.82 ALDH1A1 (0.45) ALDH1A1HPGDRAB9ANPC1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8674113-B2 Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-03-18 US disclosed
US-20120149676-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149676-A1 NOVEL COMPOUNDS PTGS1, PTGER1, PTGES ALDH1A1 126/4885HPGD 20/4885RAB9A 1033/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.