SCHEMBL9944736

SCHEMBL9944736

CNc1cc(F)c(C(=O)N[C@H]2CC[C@H](C)CC2)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
TAS1R3 Q7RTX0 3/20 0.43
TAS1R1 Q7RTX1 3/20 0.43
TAS1R2 Q8TE23 3/20 0.43
HPGD P15428 1/20 0.41
CNR1 P21554 3/20 0.40
CNR2 P34972 3/20 0.40
HCAR3 P49019 2/20 0.38
CDC25B P30305 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1727200 0.88 ALDH1A1 (0.45) ALDH1A1TAS1R3TAS1R1TAS1R2HPGD
SCHEMBL1727199 0.88 ALDH1A1 (0.45) ALDH1A1TAS1R3TAS1R1TAS1R2HPGD
SCHEMBL9944747 0.86 ALDH1A1 (0.53) ALDH1A1RAB9ANPC1TAS1R3TAS1R1
SCHEMBL9945003 0.86 ALDH1A1 (0.53) ALDH1A1RAB9ANPC1TAS1R3TAS1R1
SCHEMBL11992707 0.85 ALDH1A1 (0.48) ALDH1A1RAB9ANPC1TAS1R3TAS1R1
SCHEMBL9944827 0.84 KDM1A (0.40) ALDH1A1HPGDHCAR3CDC25B
SCHEMBL9944905 0.82 ALDH1A1 (0.44) ALDH1A1RAB9ANPC1TAS1R3TAS1R1
SCHEMBL9944735 0.82 ALDH1A1 (0.42) ALDH1A1RAB9ANPC1TAS1R3TAS1R1
SCHEMBL9944825 0.82 POLB (0.44) ALDH1A1RAB9ANPC1POLB
SCHEMBL9944914 0.82 ALDH1A1 (0.42) ALDH1A1RAB9ANPC1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8759537-B2 3H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-06-24 US disclosed
US-8674113-B2 Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-03-18 US disclosed
US-20120214786-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-23 US disclosed
US-20120149676-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149676-A1 NOVEL COMPOUNDS PTGS1, PTGER1, PTGES ALDH1A1 126/4885RAB9A 1033/4885NPC1 1695/4885
US-20120214786-A1 NEW COMPOUNDS PTGER1, PTGS1, PTGES ALDH1A1 184/4885RAB9A 2718/4885NPC1 741/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.