SCHEMBL9947008

SCHEMBL9947008

CNc1cc(N2CCN(C3CC3)CC2)c(C(=O)NC2CCC(C(F)(F)F)CC2)cc1N

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGES O14684 17/20 0.46
DRD2 P14416 3/20 0.37
ADRA1D P25100 3/20 0.37
ADRA1A P35348 3/20 0.37
ADRA1B P35368 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9946728 1.00 PTGES (0.46) PTGESDRD2ADRA1DADRA1AADRA1B
SCHEMBL9946720 0.91 PTGES (0.44) PTGES
SCHEMBL9946615 0.90 PTGES (0.43) PTGES
SCHEMBL9946574 0.90 PTGES (0.46) PTGES
SCHEMBL9944932 0.89 RAB9A (0.40) PTGESDRD2ADRA1DADRA1AADRA1B
SCHEMBL9946870 0.88 PTGES (0.46) PTGES
SCHEMBL9947062 0.88 PTGES (0.39) PTGES
SCHEMBL9946649 0.88 PTGES (0.39) PTGES
SCHEMBL9947032 0.88 PTGES (0.46) PTGES
SCHEMBL9946586 0.88 PTGES (0.48) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076673-A1 6-AMINO-2-PHENYLAMINO-1H-BENZIMIDAZOLE-5-CARBOXAMIDE- DERIVATIVES AND THEIR USE AS MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed