SCHEMBL9947032

SCHEMBL9947032

CNc1cc(N2CCOCC2)c(C(=O)NC2CCC(C(F)(F)F)CC2)cc1N

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGES O14684 12/20 0.46
ALDH1A1 P00352 1/20 0.41
USP30 Q70CQ3 1/20 0.40
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
BMPR1B O00238 1/20 0.39
BMPR1A P36894 1/20 0.39
TGFBR1 P36897 1/20 0.39
ACVRL1 P37023 1/20 0.39
ACVR1 Q04771 1/20 0.39
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
TYK2 P29597 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9946870 1.00 PTGES (0.46) PTGESALDH1A1USP30LMNATSHR
SCHEMBL9946574 0.92 PTGES (0.46) PTGES
SCHEMBL9946720 0.91 PTGES (0.44) PTGESALDH1A1
SCHEMBL9946615 0.88 PTGES (0.43) PTGES
SCHEMBL9947008 0.88 PTGES (0.46) PTGES
SCHEMBL9946649 0.88 PTGES (0.39) PTGES
SCHEMBL9947062 0.88 PTGES (0.39) PTGES
SCHEMBL9946728 0.88 PTGES (0.46) PTGES
SCHEMBL9944987 0.88 ALDH1A1 (0.44) ALDH1A1USP30LMNATSHRHTT
SCHEMBL16300080 0.87 PTGES (0.43) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076673-A1 6-AMINO-2-PHENYLAMINO-1H-BENZIMIDAZOLE-5-CARBOXAMIDE- DERIVATIVES AND THEIR USE AS MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed