SCHEMBL9947560

SCHEMBL9947560

Cc1ccc(-c2nnn(C)c2-c2cn(-c3ccc(C(=O)NC4(C)COC4)cn3)cn2)cc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 3/20 0.40
ABL1 P00519 5/20 0.38
EGLN1 Q9GZT9 4/20 0.36
WNT1 P04628 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
HDAC1 Q13547 3/20 0.34
KCNH2 Q12809 1/20 0.33
GAA P10253 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
GABRA1 P14867 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9895436 0.93 GABRA5 (0.42) GABRA5ABL1EGLN1HDAC1KCNH2
SCHEMBL9895679 0.85 GABRA5 (0.37) GABRA5ABL1EGLN1CYP1A2
SCHEMBL9947565 0.83 GABRA5 (0.42) GABRA5EGLN1GAA
SCHEMBL9895619 0.82 GABRA5 (0.47) GABRA5ABL1CYP1A2
SCHEMBL9947559 0.81 MAP4K4 (0.39) DYRK1A
SCHEMBL9894886 0.76 GABRA5 (0.51) GABRA5ABL1CYP1A2CYP2C19
SCHEMBL9895606 0.76 EGLN1 (0.40) GABRA5EGLN1HDAC1GABRA1
SCHEMBL9895449 0.76 GABRA5 (0.53) GABRA5EGLN1
SCHEMBL9894488 0.75 GABRA5 (0.43) GABRA5EGLN1CYP1A2CYP2C19
SCHEMBL9895824 0.75 GABRA5 (0.39) GABRA5ABL1HDAC1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076590-A1 NOVEL TRIAZOLE COMPOUNDS III F. HOFFMANN-LA ROCHE AG (CH) 2012-06-14 WO disclosed