SCHEMBL9947565

SCHEMBL9947565

Cc1ccc(-c2nnn(C)c2-c2cn(-c3ccc(C(=O)NC(C)C)cn3)cn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 12/20 0.42
CNR1 P21554 1/20 0.41
EGLN1 Q9GZT9 4/20 0.40
GRM1 Q13255 1/20 0.40
GAA P10253 1/20 0.35
PHGDH O43175 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9894488 0.92 GABRA5 (0.43) GABRA5EGLN1GRM1
SCHEMBL9947559 0.86 MAP4K4 (0.39)
SCHEMBL9895430 0.83 GABRA5 (0.44) GABRA5EGLN1
SCHEMBL9947560 0.83 GABRA5 (0.40) GABRA5EGLN1GAA
SCHEMBL9894510 0.80 RAB9A (0.42) GABRA5
SCHEMBL9894907 0.80 GABRA5 (0.44) GABRA5GRM1PHGDH
SCHEMBL27933840 0.78 KDM4C (0.42) GABRA5
SCHEMBL6468600 0.77 GABRA5 (0.49) GABRA5GRM1
SCHEMBL9895449 0.75 GABRA5 (0.53) GABRA5EGLN1
SCHEMBL9895133 0.74 GABRA5 (0.43) GABRA5EGLN1GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076590-A1 NOVEL TRIAZOLE COMPOUNDS III F. HOFFMANN-LA ROCHE AG (CH) 2012-06-14 WO disclosed