SCHEMBL9947559

SCHEMBL9947559

Cc1ccc(-c2nnn(C)c2-c2cn(-c3ccc(C(N)=O)cn3)cn2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.39
F9 P00740 1/20 0.36
KDR P35968 1/20 0.36
MAPK1 P28482 1/20 0.35
MAP2K4 P45985 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
MAPKAPK3 Q16644 1/20 0.35
MAPK6 Q16659 1/20 0.35
MAPKAPK5 Q8IW41 1/20 0.35
HSP90AA1 P07900 3/20 0.35
KDM2B Q8NHM5 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM1A O60341 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
CPB2 Q96IY4 3/20 0.33
SRC P12931 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9895465 0.91 TNIK (0.41) MAP4K4DYRK1A
SCHEMBL9947565 0.86 GABRA5 (0.42)
SCHEMBL27933840 0.82 KDM4C (0.42) MAP4K4KDM4C
SCHEMBL9895366 0.82 MAP4K4 (0.37) MAP4K4HSP90AA1DYRK1A
SCHEMBL9895921 0.82 HTR5A (0.36) MAP4K4HSP90AA1DYRK1A
SCHEMBL9947560 0.81 GABRA5 (0.40) DYRK1A
SCHEMBL9895019 0.78 MAP4K4 (0.53) MAP4K4KDM4CP2RY14
SCHEMBL9894488 0.78 GABRA5 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9895436 0.74 GABRA5 (0.42)
SCHEMBL9895449 0.73 GABRA5 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076590-A1 NOVEL TRIAZOLE COMPOUNDS III F. HOFFMANN-LA ROCHE AG (CH) 2012-06-14 WO disclosed