SCHEMBL9947652

SCHEMBL9947652

Cc1c(C(=O)O)c(C)n(-c2ccccc2)c(=O)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
GFER P55789 1/20 0.47
ALDH1A1 P00352 3/20 0.44
NOTUM Q6P988 3/20 0.44
KDM4E B2RXH2 3/20 0.44
MAPT P10636 1/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
PTGFR P43088 1/20 0.42
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11457576 0.89 ALDH1A1 (0.43) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL11468129 0.87 NOTUM (0.48) ALDH1A1NOTUMKDM4EL3MBTL1PTGFR
SCHEMBL11464864 0.87 NOTUM (0.48) GAAALDH1A1NOTUMKDM4EMAPT
SCHEMBL2035472 0.85 GAA (0.50) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9948181 0.83 GAA (0.48) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947636 0.82 TAAR1 (0.47) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947581 0.81 NOTUM (0.47) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947824 0.81 GAA (0.47) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947765 0.80 TAAR1 (0.48) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947980 0.79 TAAR1 (0.46) GAAGFERALDH1A1NOTUMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP claimed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US claimed
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP disclosed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US disclosed