SCHEMBL9947980

SCHEMBL9947980

CCc1c(C)c(C(=O)O)c(C)n(-c2ccccc2)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.46
GAA P10253 1/20 0.45
GFER P55789 1/20 0.45
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 3/20 0.43
RECQL P46063 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
POLB P06746 2/20 0.43
HTT P42858 1/20 0.42
NOTUM Q6P988 1/20 0.42
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 2/20 0.41
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9947669 0.84 MEN1 (0.49) TAAR1GAAGFERMEN1KMT2A
SCHEMBL9947636 0.83 TAAR1 (0.47) TAAR1GAAGFERMEN1KMT2A
SCHEMBL2035472 0.83 GAA (0.50) TAAR1GAAGFERMEN1KMT2A
SCHEMBL9948181 0.80 GAA (0.48) TAAR1GAAGFERMEN1KMT2A
SCHEMBL9947824 0.79 GAA (0.47) TAAR1GAAGFERMEN1KMT2A
SCHEMBL9947652 0.79 GAA (0.47) TAAR1GAAGFERMEN1KMT2A
SCHEMBL23147061 0.77 NOTUM (0.47) TAAR1KDM4EALDH1A1SMN1; SMN2POLB
Hydrochloric Acid SCHEMBL29971235 0.76 NOTUM (0.46) TAAR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL9947638 0.76 MEN1 (0.50) TAAR1GAAGFERMEN1KMT2A
SCHEMBL9947711 0.75 KDM4E (0.54) GAAGFERMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP claimed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US claimed
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP disclosed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US disclosed