SCHEMBL9948181

SCHEMBL9948181

Cc1c(C(=O)O)c(C)n(-c2ccccc2)c(=O)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
GFER P55789 1/20 0.48
ALDH1A1 P00352 3/20 0.45
NOTUM Q6P988 2/20 0.45
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 1/20 0.44
ATM Q13315 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
PKM P14618 1/20 0.43
HKDC1 Q2TB90 1/20 0.43
RORC P51449 1/20 0.42
KAT2B Q92831 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2035472 0.87 GAA (0.50) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947652 0.83 GAA (0.47) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947824 0.83 GAA (0.47) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947669 0.82 MEN1 (0.49) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947806 0.81 NOTUM (0.48) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947980 0.80 TAAR1 (0.46) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL9947638 0.80 MEN1 (0.50) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL11456551 0.79 NOTUM (0.51) GAAALDH1A1NOTUMKDM4EMEN1
SCHEMBL9947711 0.79 KDM4E (0.54) GAAGFERALDH1A1NOTUMKDM4E
SCHEMBL2014199 0.79 GAA (0.44) GAAGFERALDH1A1NOTUMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP claimed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US claimed
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP disclosed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US disclosed