SCHEMBL9947711

SCHEMBL9947711

Cc1c(C(=O)O)c(C)n(-c2ccccc2)c(=O)c1C#N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.54
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
HPGD P15428 1/20 0.49
ALDH1A1 P00352 5/20 0.46
RXFP1 Q9HBX9 1/20 0.46
ALOX15 P16050 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GAA P10253 1/20 0.44
GFER P55789 1/20 0.44
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
NOTUM Q6P988 1/20 0.41
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014199 0.86 GAA (0.44) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL2035472 0.82 GAA (0.50) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL9947695 0.81 GAA (0.43) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL9948181 0.79 GAA (0.48) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL23146873 0.78 KDM4E (0.52) KDM4EHPGDALDH1A1HSD17B10GAA
SCHEMBL14138730 0.78 HPGD (0.52) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL9947652 0.78 GAA (0.47) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL9947824 0.78 GAA (0.47) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL9947980 0.75 TAAR1 (0.46) KDM4ECYP1A2CYP2C9HPGDALDH1A1
SCHEMBL1718143 0.75 GAA (0.45) KDM4EHPGDALDH1A1GAAGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP claimed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US claimed
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP disclosed
US-8207347-B2 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2012-06-26 US disclosed