SCHEMBL9952090

SCHEMBL9952090

COc1c(Br)cc(Cl)cc1CC=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
CYP1A2 P05177 3/20 0.39
CYP2D6 P10635 2/20 0.39
MEN1 O00255 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.38
CA2 P00918 2/20 0.37
CA4 P22748 2/20 0.37
IMPDH2 P12268 2/20 0.37
ERN1 O75460 2/20 0.36
CA1 P00915 1/20 0.36
CA6 P23280 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14612683 0.84 CA2 (0.41) KMT2ACYP1A2CYP2D6MEN1SMN1; SMN2
SCHEMBL8427155 0.82 KMT2A (0.54) KMT2ACYP1A2CYP2D6MEN1SMN1; SMN2
SCHEMBL5272430 0.81 ALDH1A1 (0.46) KMT2ACYP1A2CYP2D6MEN1SMN1; SMN2
SCHEMBL4932262 0.79 KMT2A (0.46) KMT2ACYP1A2CYP2D6MEN1SMN1; SMN2
SCHEMBL21198098 0.77 THRB (0.47) KMT2ACYP1A2CYP2D6MEN1SMN1; SMN2
SCHEMBL30930936 0.77 CA2 (0.52) KMT2AMEN1SMN1; SMN2CA2CA4
SCHEMBL9952803 0.76 TAAR1 (0.49) KMT2ACYP1A2MEN1SMN1; SMN2CA2
SCHEMBL4021512 0.75 ERN1 (0.55) KMT2ACYP1A2MEN1CYP2C9CYP2C19
SCHEMBL2389960 0.75 ERN1 (0.55) CYP1A2CYP2C19CA2CA4ERN1
SCHEMBL10265435 0.75 KMT2A (0.50) KMT2ACYP1A2CYP2D6MEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP disclosed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO disclosed