SCHEMBL9953247

SCHEMBL9953247

COc1c(CCOC(N)=O)cc(Cl)c(C)c1-c1cccc(C(=O)N(C)C)n1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 13/20 0.36
CD274 Q9NZQ7 2/20 0.34
PDCD1LG2 Q9BQ51 1/20 0.34
PDCD1 Q15116 1/20 0.32
CTSA P10619 1/20 0.32
F10 P00742 2/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953244 0.89 PIK3CD (0.37) PIK3CDCTSAHCRTR1HCRTR2
SCHEMBL9952249 0.84 HCRTR1 (0.38) PIK3CDCTSAHCRTR1HCRTR2
SCHEMBL9929633 0.78 PIK3CD (0.47) PIK3CDCD274PDCD1LG2
Hydrochloric Acid SCHEMBL9929471 0.77 PIK3CD (0.46) PIK3CDCD274PDCD1LG2CTSA
SCHEMBL9952247 0.74 PIK3CD (0.46) PIK3CDCTSA
SCHEMBL9929037 0.71 PIK3CD (0.41) PIK3CDCTSA
SCHEMBL9952278 0.71 ALDH1A1 (0.38) CD274PDCD1LG2
SCHEMBL9952356 0.69 NQO2 (0.43)
SCHEMBL9952282 0.69 NQO2 (0.43)
SCHEMBL28712872 0.69 ALDH1A1 (0.44) CD274PDCD1LG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP disclosed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO disclosed