SCHEMBL9952249

SCHEMBL9952249

COc1c(CCNC(=O)O)cc(Cl)c(C)c1-c1cccc(C(=O)N(C)C)n1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
CTSA P10619 2/20 0.35
SLC2A1 P11166 1/20 0.35
PIK3CD O00329 8/20 0.34
MTNR1A P48039 2/20 0.34
MTNR1B P49286 2/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
PTGDR Q13258 1/20 0.33
P2RX7 Q99572 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
APLNR P35414 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953244 0.87 PIK3CD (0.37) HCRTR1HCRTR2CTSAPIK3CDAPLNR
SCHEMBL9953247 0.84 PIK3CD (0.36) HCRTR1HCRTR2CTSAPIK3CD
SCHEMBL9952282 0.81 NQO2 (0.43) KDM4ELMNAPTGDRALDH1A1HPGD
SCHEMBL9952356 0.79 NQO2 (0.43) KDM4ELMNAPTGDRALDH1A1HPGD
SCHEMBL9952247 0.78 PIK3CD (0.46) CTSAPIK3CDAPLNR
SCHEMBL9929633 0.77 PIK3CD (0.47) PIK3CD
Hydrochloric Acid SCHEMBL9929471 0.76 PIK3CD (0.46) CTSAPIK3CD
SCHEMBL9929037 0.73 PIK3CD (0.41) CTSAPIK3CDAPLNRCNR2
SCHEMBL9952889 0.73 CYP1A2 (0.45) HPGD
SCHEMBL9952473 0.70 IMPDH2 (0.41) SLC2A1MTNR1AMTNR1BKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP disclosed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO disclosed