SCHEMBL9953743

SCHEMBL9953743

COc1ncc(Br)cc1C(=N)NO

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.34
OPRK1 P41145 14/20 0.34
HSD17B10 Q99714 1/20 0.33
PIK3C3 Q8NEB9 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
ALOX12 P18054 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
AURKA O14965 1/20 0.31
TTK P33981 1/20 0.31
AURKB Q96GD4 1/20 0.31
INCENP Q9NQS7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764171 0.85 CNR2 (0.35) CNR2OPRK1NPC1RAB9AALDH1A1
SCHEMBL757419 0.78 OPRK1 (0.49) OPRK1HSD17B10
SCHEMBL29457453 0.78 OPRK1 (0.49) OPRK1HSD17B10
SCHEMBL14764185 0.76 HTT (0.44) CNR2OPRK1HSD17B10PIK3C3NPC1
SCHEMBL316314 0.76 HSD17B10 (0.50) CNR2OPRK1HSD17B10ALDH1A1
SCHEMBL29527502 0.75 OPRK1 (0.44) CNR2OPRK1HSD17B10NPC1RAB9A
SCHEMBL839912 0.75 OPRK1 (0.44) CNR2OPRK1HSD17B10NPC1RAB9A
SCHEMBL11875941 0.75 CNR2 (0.38) CNR2OPRK1HSD17B10NPC1RAB9A
SCHEMBL9953358 0.75 ALDH1A1 (0.38) CNR2OPRK1ALDH1A1MAPTAURKA
Lithium SCHEMBL9954426 0.75 HSD17B10 (0.49) CNR2OPRK1HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed