SCHEMBL9954016

SCHEMBL9954016

COc1ncc(Br)cc1S(=O)(=O)N1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
HTT P42858 2/20 0.48
KDM4E B2RXH2 3/20 0.48
LMNA P02545 1/20 0.48
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
KMT2A Q03164 2/20 0.46
NPC1 O15118 1/20 0.45
GAA P10253 1/20 0.45
HSD17B10 Q99714 2/20 0.44
CASP1 P29466 1/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789757 0.88 GAA (0.58) TSHRKDM4ELMNAALDH1A1NPSR1
SCHEMBL14305917 0.86 GAA (0.57) TSHRKDM4ELMNAALDH1A1NPSR1
SCHEMBL10289141 0.85 MAPT (0.49) TSHRKDM4ELMNAALDH1A1GAA
SCHEMBL28096087 0.82 HSD17B10 (0.52) TSHRKDM4ELMNAALDH1A1KMT2A
SCHEMBL730137 0.80 KDM4E (0.58) KDM4EKMT2ANPC1HSD17B10MEN1
SCHEMBL9954366 0.78 ALPL (0.50) TSHRHTTKDM4ELMNAALDH1A1
SCHEMBL9955070 0.78 GAA (0.41) TSHRKDM4EALDH1A1NPSR1KMT2A
SCHEMBL9954790 0.77 SHMT2 (0.41) TSHRHTTKDM4ELMNAALDH1A1
SCHEMBL15052436 0.76 GAA (0.77) TSHRKDM4ELMNAALDH1A1NPSR1
SCHEMBL9953196 0.73 PIK3CG (0.46) HTTKDM4EKMT2AHSD17B10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed