SCHEMBL28096087

SCHEMBL28096087

CCN1CCN(S(=O)(=O)c2cc(Br)cnc2OC)CC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.52
MAPK1 P28482 1/20 0.52
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
TSHR P16473 1/20 0.50
KMT2A Q03164 2/20 0.48
CYP2D6 P10635 1/20 0.44
GAA P10253 2/20 0.43
TNF P01375 2/20 0.42
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10289141 0.86 MAPT (0.49) HSD17B10MAPK1ALDH1A1KDM4ETSHR
SCHEMBL789757 0.85 GAA (0.58) HSD17B10ALDH1A1KDM4ETSHRKMT2A
SCHEMBL14305917 0.84 GAA (0.57) HSD17B10ALDH1A1KDM4ETSHRKMT2A
SCHEMBL9954016 0.82 TSHR (0.50) HSD17B10ALDH1A1KDM4ETSHRKMT2A
SCHEMBL9955070 0.76 GAA (0.41) HSD17B10ALDH1A1KDM4ETSHRKMT2A
SCHEMBL9954790 0.75 SHMT2 (0.41) HSD17B10ALDH1A1KDM4ETSHRKMT2A
SCHEMBL2402633 0.72 ALDH1A1 (0.70) ALDH1A1KDM4ETSHRKMT2ACYP2D6
SCHEMBL6200528 0.72 KMT2A (0.83) HSD17B10MAPK1ALDH1A1KDM4ETSHR
SCHEMBL2379664 0.72 ALDH1A1 (0.62) HSD17B10MAPK1ALDH1A1KDM4ETSHR
SCHEMBL6447545 0.71 ALDH1A1 (0.64) ALDH1A1TSHRKMT2ACYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104011045-B Dihydrobenzoxazine and dihydropyridinooxazine derivatives 诺华股份有限公司 2016-08-24 CN disclosed