SCHEMBL9954342

SCHEMBL9954342

N#Cc1cccc(Nc2ncc3c(n2)CCNC3)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.58
GRM5 P41594 2/20 0.58
SYK P43405 2/20 0.54
CDK5 Q00535 6/20 0.48
CDK5R1 Q15078 6/20 0.48
CDK2 P24941 6/20 0.48
CCNA2 P20248 4/20 0.48
CDK1 P06493 2/20 0.48
CCNB1 P14635 2/20 0.48
CDC7 O00311 1/20 0.48
IGF1R P08069 1/20 0.46
IKBKE Q14164 1/20 0.45
CDK4 P11802 2/20 0.44
CCNT1 O60563 1/20 0.44
CCNE1 P24864 1/20 0.44
CCND3 P30281 1/20 0.44
FLT3 P36888 1/20 0.44
CDK9 P50750 1/20 0.44
CDK6 Q00534 1/20 0.44
JAK1 P23458 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9958931 0.83 GRM5 (0.55) MAOBGRM5CDK5CDK5R1CDK2
SCHEMBL9958935 0.83 GRM5 (0.70) MAOBGRM5SYKCDK5CDK5R1
SCHEMBL9959907 0.83 CDK5 (0.70) MAOBGRM5CDK5CDK5R1CDK2
SCHEMBL17620607 0.82 CDK5 (0.65) MAOBGRM5CDK5CDK5R1CDK2
SCHEMBL19475557 0.81 GRM5 (0.56) MAOBGRM5SYKCDK5CDK5R1
SCHEMBL9959330 0.81 CDK5 (0.71) MAOBGRM5SYKCDK5CDK5R1
SCHEMBL30099826 0.77 GRM5 (0.53) MAOBGRM5SYKCDK5CDK5R1
SCHEMBL9955805 0.76 PDGFRB (0.56) MAOBGRM5SYKJAK3EGFR
SCHEMBL22999621 0.75 CDK5 (0.51) CDK5CDK5R1CDK2CCNA2CDK1
SCHEMBL9959904 0.75 CDK2 (0.67) MAOBGRM5CDK5CDK5R1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085167-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed