SCHEMBL9955265

SCHEMBL9955265

COCCn1c(N)nc2ccc(Br)cc2c1=O.COCCn1c(NC#N)nc2ccc(Br)cc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.41
ALDH1A1 P00352 10/20 0.37
CYP1A2 P05177 6/20 0.36
CYP2D6 P10635 3/20 0.36
CASP1 P29466 3/20 0.36
CASP7 P55210 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 5/20 0.36
KDM4E B2RXH2 4/20 0.36
GAA P10253 3/20 0.36
GLA P06280 2/20 0.36
TSHR P16473 2/20 0.36
USP2 O75604 2/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
CASP3 P42574 2/20 0.35
CYP2C9 P11712 3/20 0.35
MAPT P10636 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954047 0.91 HSD17B10 (0.41) HSD17B10ALDH1A1CYP1A2CYP2D6CASP1
SCHEMBL9953325 0.87 HSD17B10 (0.49) HSD17B10ALDH1A1CYP1A2CYP2D6CASP1
SCHEMBL10289053 0.82 KDM4E (0.50) HSD17B10ALDH1A1CYP1A2CASP1CASP7
SCHEMBL31241102 0.82 CACNA2D1 (0.42) ALDH1A1MEN1KMT2AKDM4EUSP2
SCHEMBL31241091 0.75 CACNA2D1 (0.47) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL9954454 0.73 MEN1 (0.41) HSD17B10ALDH1A1CYP1A2CYP2D6CASP1
SCHEMBL9954050 0.72 HSD17B10 (0.41) HSD17B10ALDH1A1CYP1A2CYP2D6CASP1
SCHEMBL10289136 0.72 CACNA2D1 (0.51) CYP1A2CYP2D6MEN1KMT2ACASP3
SCHEMBL9955108 0.71 MEN1 (0.40) ALDH1A1MEN1KMT2ACYP3A4GAA
SCHEMBL9954166 0.71 ALDH1A1 (0.42) HSD17B10ALDH1A1CASP1CASP7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed