SCHEMBL9956153

SCHEMBL9956153

Cc1ccn(-c2ccccc2C(=O)O)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 4/20 0.53
NR4A1 P22736 1/20 0.53
ALDH1A1 P00352 3/20 0.50
MAPT P10636 3/20 0.50
RAB9A P51151 2/20 0.50
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
TSHR P16473 1/20 0.49
ALOX15 P16050 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
POLB P06746 2/20 0.46
APEX1 P27695 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NOTUM Q6P988 1/20 0.44
NPC1 O15118 1/20 0.43
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTT P42858 1/20 0.43
AKR1C3 P42330 2/20 0.43
AKR1C2 P52895 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16573945 0.81 MAPT (0.45) ALDH1A1MAPTRAB9AKDM4EGAA
SCHEMBL9956115 0.81 KDM4E (0.51) MYCNR4A1ALDH1A1MAPTRAB9A
SCHEMBL23981879 0.78 MAPT (0.49) MYCALDH1A1MAPTRAB9AKDM4E
SCHEMBL4450463 0.75 GAA (0.67) ALDH1A1MAPTRAB9AKDM4EGAA
SCHEMBL31316722 0.75 F2 (0.51) MYCNR4A1ALDH1A1MAPTKDM4E
SCHEMBL10262760 0.74 ALDH1A1 (0.55) ALDH1A1MAPTRAB9AKDM4EGAA
SCHEMBL25254882 0.74 HTT (0.56) ALDH1A1MAPTRAB9AKDM4EGAA
SCHEMBL1339393 0.72 ALDH1A1 (0.50) MYCNR4A1ALDH1A1MAPTKDM4E
SCHEMBL17256244 0.72 MYC (0.51) MYCNR4A1ALDH1A1MAPTTSHR
SCHEMBL31525258 0.72 RAB9A (0.43) ALDH1A1MAPTRAB9AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
CN-1391476-A Vasopressin agonist formulation and process AMERICAN CYANAMID CO (US) 2003-01-15 CN disclosed