SCHEMBL9956338

SCHEMBL9956338

Cc1n[c]oc1-c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
GAA P10253 2/20 0.39
L3MBTL1 Q9Y468 3/20 0.37
MEN1 O00255 2/20 0.37
NFKB1 P19838 2/20 0.37
NFKB2 Q00653 2/20 0.37
KMT2A Q03164 2/20 0.37
RELA Q04206 2/20 0.37
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
NOTUM Q6P988 2/20 0.37
MBNL1 Q9NR56 1/20 0.37
DCUN1D1 Q96GG9 2/20 0.36
ACHE P22303 1/20 0.35
ALDH1A1 P00352 2/20 0.35
PKM P14618 2/20 0.35
NMUR2 Q9GZQ4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4511404 0.75 BRD4 (0.38) NPC1RAB9ASMN1; SMN2L3MBTL1MEN1
SCHEMBL10263295 0.70 NPC1 (0.42) NPC1RAB9ASMN1; SMN2GAAL3MBTL1
SCHEMBL9955370 0.70 NOTUM (0.44) NPC1RAB9ASMN1; SMN2GAAL3MBTL1
SCHEMBL9955349 0.70 NOTUM (0.39) SMN1; SMN2GAAL3MBTL1MGAMSI
SCHEMBL558381 0.68 KDM4E (0.36) NPC1RAB9ASMN1; SMN2GAAL3MBTL1
SCHEMBL13960109 0.68 NPC1 (0.44) NPC1RAB9ASMN1; SMN2GAAL3MBTL1
SCHEMBL14112980 0.68 NPC1 (0.41) NPC1RAB9ASMN1; SMN2GAAL3MBTL1
SCHEMBL9954602 0.68 NPC1 (0.41) NPC1RAB9ASMN1; SMN2GAAL3MBTL1
SCHEMBL29001802 0.67 MEN1 (0.36) NPC1RAB9ASMN1; SMN2L3MBTL1MEN1
SCHEMBL9956367 0.66 RAB9A (0.42) NPC1RAB9ASMN1; SMN2GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed