SCHEMBL9956367

SCHEMBL9956367

Cc1cccc(-c2o[c]nc2C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.42
NPC1 O15118 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 4/20 0.38
POLB P06746 2/20 0.38
TP53 P04637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ENPP3 O14638 1/20 0.38
NOTUM Q6P988 1/20 0.38
ACHE P22303 1/20 0.38
CASP3 P42574 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
GAA P10253 2/20 0.38
IDO1 P14902 1/20 0.38
METAP2 P50579 1/20 0.38
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955349 0.83 NOTUM (0.39) SMN1; SMN2TP53NOTUMACHEGAA
SCHEMBL9955323 0.83 ESR2 (0.44) RAB9ANPC1SMN1; SMN2TSHRALDH1A1
SCHEMBL9956334 0.69 IMPDH2 (0.56) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL5548164 0.69 RAB9A (0.49) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL7948113 0.69 RAB9A (0.47) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL29373699 0.68 ACHE (0.69) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL31471473 0.68 ACHE (0.69) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL301247 0.68 ACHE (0.69) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL9956286 0.68 ENPP3 (0.45) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL8626847 0.68 RAB9A (0.54) RAB9ANPC1SMN1; SMN2HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed