SCHEMBL9956636

SCHEMBL9956636

O=C(O)N1CC2CCN(c3cnc4c(F)c(F)ccc4n3)CC21

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.38
DPP8 Q6V1X1 2/20 0.38
DPP7 Q9UHL4 2/20 0.38
DPP9 Q86TI2 1/20 0.38
HCRTR1 O43613 11/20 0.36
HCRTR2 O43614 11/20 0.36
JAK3 P52333 5/20 0.34
LCK P06239 1/20 0.34
BTK Q06187 1/20 0.34
PARP1 P09874 1/20 0.34
CCR4 P51679 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9956083 0.92 DPP4 (0.38) DPP4DPP8DPP7DPP9HCRTR1
SCHEMBL9957137 0.88 HCRTR1 (0.44) DPP4DPP8DPP7DPP9HCRTR1
SCHEMBL9957734 0.86 RET (0.42)
SCHEMBL9957737 0.86 RET (0.42)
SCHEMBL9958187 0.85 HCRTR1 (0.45) DPP4DPP8DPP7DPP9HCRTR1
SCHEMBL9957907 0.84 HCRTR1 (0.44) DPP4DPP8DPP7DPP9HCRTR1
SCHEMBL9958172 0.82 HCRTR1 (0.44) DPP4DPP8DPP7DPP9HCRTR1
SCHEMBL9956949 0.82 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL9957559 0.81 HCRTR1 (0.44) DPP4DPP8DPP7DPP9HCRTR1
SCHEMBL9957415 0.81 HCRTR1 (0.45) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed