SCHEMBL9958172

SCHEMBL9958172

O=C(O)N1CC2CCN(c3cnc4ccc(F)cc4n3)CC21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.44
HCRTR2 O43614 12/20 0.44
DPP4 P27487 1/20 0.42
DPP8 Q6V1X1 1/20 0.42
DPP9 Q86TI2 1/20 0.42
DPP7 Q9UHL4 1/20 0.42
PIK3CA P42336 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
DGAT1 O75907 1/20 0.38
ADORA2A P29274 1/20 0.38
KCNH2 Q12809 1/20 0.38
PDE10A Q9Y233 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9957907 0.96 HCRTR1 (0.44) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9958187 0.88 HCRTR1 (0.45) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9957542 0.85 HCRTR1 (0.50) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9956636 0.82 DPP4 (0.38) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9956083 0.82 DPP4 (0.38) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9957068 0.81 RET (0.46) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9957065 0.81 RET (0.46) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9957137 0.80 HCRTR1 (0.44) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9957559 0.80 HCRTR1 (0.44) HCRTR1HCRTR2DPP4DPP8DPP9
SCHEMBL9957037 0.78 HCRTR1 (0.45) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed