SCHEMBL9958613

SCHEMBL9958613

Cc1nc(-c2cccc(-c3cnc(N)nc3)c2)ncc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
CLK1 P49759 2/20 0.41
ALOX5AP P20292 8/20 0.40
FEN1 P39748 6/20 0.40
MAP4K4 O95819 2/20 0.40
PIK3CB P42338 1/20 0.40
DHFR P00374 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3569775 0.80 MAP4K4 (0.41) ADORA2AADORA1ALOX5APFEN1MAP4K4
SCHEMBL9957837 0.78 KIF18A (0.47) ALOX5APFEN1
SCHEMBL3571995 0.75 DHODH (0.42) ADORA2AADORA1ALOX5APFEN1MAP4K4
SCHEMBL5327094 0.75 ADORA1 (0.69) ADORA2AADORA1DHFR
SCHEMBL9958759 0.74 LRRK2 (0.44)
SCHEMBL5318644 0.72 ADORA2A (0.60) ADORA2AADORA1ALOX5APFEN1MAP4K4
SCHEMBL29818212 0.72 KIF11 (0.59) CLK1ALOX5APFEN1MAP4K4
SCHEMBL3570340 0.71 MAP4K4 (0.46) ADORA2AADORA1ALOX5APFEN1MAP4K4
SCHEMBL3569085 0.70 ALOX5AP (0.41) ADORA2AADORA1CLK1ALOX5APFEN1
SCHEMBL3562521 0.70 MAP4K4 (0.45) MAP4K4PIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468727-A1 Pyridine and pyrimidine derivatives as MGLUR2 antagonists F. Hoffmann-La Roche AG (CH) 2012-06-27 EP claimed