SCHEMBL9959772

SCHEMBL9959772

CC(C)CNC(CC(N)=O)c1cn(C)cn1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 6/20 0.38
CPB1 P15086 4/20 0.35
CPA1 P15085 1/20 0.32
FPR1 P21462 1/20 0.31
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
MTOR P42345 1/20 0.30
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30
DCAF1 Q9Y4B6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8843361 0.99 CPB2 (0.37) CPB2CPB1CPA1FPR1
Hydrochloric Acid SCHEMBL8844341 0.79 LMNA (0.43) CPB2DCAF1
Hydrochloric Acid SCHEMBL8340839 0.77 SYK (0.37) CPB2HTT
Hydrochloric Acid SCHEMBL8844102 0.71 MEN1 (0.45) TSHRGAA
SCHEMBL9953903 0.70 CPB2 (0.43) CPB2CPB1CPA1FPR1CYP2C9
Hydrochloric Acid SCHEMBL8843356 0.69 CPB2 (0.44) CPB2CPB1CYP2C9TSHRCYP2C19
SCHEMBL3206859 0.66 CPB2 (0.46) CPB2CPB1CPA1FPR1CYP2C9
SCHEMBL5869564 0.66 CPB2 (0.46) CPB2CPB1CPA1
SCHEMBL19674649 0.65
SCHEMBL12669824 0.64 CPB2 (0.38) CPB2FPR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655330-A1 SUBSTITUTED PYRIDINES AS SODIUM CHANNEL BLOCKERS Purdue Pharma LP (US) 2013-10-30 EP disclosed
WO-2012085650-A1 SUBSTITUTED PYRIDINES AS SODIUM CHANNEL BLOCKERS PURDUE PHARMA L.P. (US) 2012-06-28 WO disclosed