SCHEMBL9963672

SCHEMBL9963672

Cc1c2nc(NCC(=O)O)sc2cc2sc(NCC(=O)N3CCCC(F)(F)C3)nc12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.38
CHRM4 P08173 1/20 0.35
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
PIK3CD O00329 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
GRM4 Q14833 2/20 0.32
DHODH Q02127 1/20 0.32
MYC P01106 1/20 0.32
WDR5 P61964 1/20 0.32
TBK1 Q9UHD2 1/20 0.31
GRM5 P41594 1/20 0.31
VNN1 O95497 1/20 0.31
FABP4 P15090 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9963654 0.91 PTGS2 (0.39) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL9963639 0.91 PTGS2 (0.44) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL9966071 0.88 PTGS2 (0.36) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL14369905 0.87 PTGS2 (0.36) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL9963695 0.87 PTGS2 (0.49) PTGS2FABP4
SCHEMBL9963641 0.87 CHRM4 (0.35) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL9963658 0.87 TP53 (0.42) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL9963607 0.87 ACHE (0.38) PTGS2CHRM4TLR9TLR8TLR7
SCHEMBL9963545 0.86 PTGS2 (0.51) PTGS2FABP4
SCHEMBL9963644 0.85 PTGS2 (0.37) PTGS2TLR9TLR8TLR7TBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8203001-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-19 US disclosed
US-8203001-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-19 US disclosed
US-20090258857-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 US disclosed
US-20090258857-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090258857-A1 CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 PTGS2 2872/4885CHRM4 820/4885TLR9 3948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.