SCHEMBL9966071

SCHEMBL9966071

Cc1c2nc(NCC(=O)N3CCCNCC3)sc2cc2sc(NCC(=O)N3CCCC(F)(F)C3)nc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.36
TLR9 Q9NR96 2/20 0.33
TLR8 Q9NR97 2/20 0.33
TLR7 Q9NYK1 2/20 0.33
CHRM4 P08173 1/20 0.33
FABP4 P15090 1/20 0.32
CCNT1 O60563 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CDK9 P50750 1/20 0.32
CCNA1 P78396 1/20 0.32
DPP4 P27487 1/20 0.32
GRM4 Q14833 2/20 0.32
PIK3CD O00329 1/20 0.31
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
DHODH Q02127 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13675181 0.91 PTGS2 (0.33) PTGS2TLR9TLR8TLR7CCNT1
SCHEMBL9963639 0.88 PTGS2 (0.44) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963672 0.88 PTGS2 (0.38) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963654 0.86 PTGS2 (0.39) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL14369905 0.85 PTGS2 (0.36) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963641 0.84 CHRM4 (0.35) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963607 0.84 ACHE (0.38) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963658 0.84 TP53 (0.42) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963660 0.83 ACHE (0.41) PTGS2TLR9TLR8TLR7CHRM4
SCHEMBL9963644 0.83 PTGS2 (0.37) PTGS2TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032583-B1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2014-11-19 EP disclosed
US-8203001-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-19 US disclosed