SCHEMBL9968002

SCHEMBL9968002

Cc1cc(S(=O)(=O)Nc2cc(I)c(I)cc2NS(=O)(=O)c2cccs2)c(C)o1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 10/20 0.54
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 1/20 0.47
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.45
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9930585 0.88 CCR2 (0.69) CCR2ALDH1A1MEN1KMT2AMAPT
SCHEMBL9968042 0.80 CCR2 (0.48) CCR2ALDH1A1MAPTTP53HPGD
SCHEMBL7590525 0.74 NPC1 (0.63) CCR2ALDH1A1KMT2ATP53HPGD
SCHEMBL9968200 0.73 CCR2 (0.62) CCR2MEN1KMT2AMAPTTP53
SCHEMBL16747597 0.71 CCR2 (0.48) CCR2ALDH1A1MEN1KMT2AMAPT
SCHEMBL9930512 0.70 CCR2 (1.00) CCR2
SCHEMBL9968068 0.70 CCR2 (0.64) CCR2MEN1KMT2A
SCHEMBL9968208 0.70 PKM (0.56) CCR2MEN1KMT2A
SCHEMBL9930712 0.69 CCR2 (0.73) CCR2MEN1KMT2AMAPTLMNA
SCHEMBL7592227 0.69 CCR2 (0.67) CCR2TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082633-A1 NOVEL 1,2- BIS-SULFONAMIDE DERIVATIVES AS CHEMOKINE RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-21 WO disclosed