SCHEMBL9970746

SCHEMBL9970746

CC(NCc1ccccc1)c1nc2ccccc2c(=O)n1-c1ccc(Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
TSHR P16473 2/20 0.48
CYP2C19 P33261 2/20 0.48
KMT2A Q03164 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
GAA P10253 1/20 0.48
CYP2D6 P10635 1/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PDE10A Q9Y233 1/20 0.47
PTGS2 P35354 1/20 0.47
JUN P05412 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL453737 0.85 SMN1; SMN2 (0.58) HTR6SMN1; SMN2ALDH1A1CYP1A2CYP3A4
SCHEMBL4582001 0.76 SMN1; SMN2 (0.56) HTR6SMN1; SMN2ALDH1A1CYP1A2CYP3A4
SCHEMBL451131 0.76 NPC1 (0.52) ALDH1A1TSHRKDM4EHPGDCXCR3
SCHEMBL12463889 0.75 PTGS2 (0.47) HTR6KMT2AMEN1PTGS2CXCR3
SCHEMBL1553514 0.75 HRH3 (0.55) SMN1; SMN2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL1664204 0.74 TRPV1 (0.47) HTR6SMN1; SMN2KMT2AMEN1JUN
SCHEMBL450858 0.74 SMN1; SMN2 (0.57) SMN1; SMN2ALDH1A1KMT2ANPSR1MEN1
SCHEMBL13291361 0.74 CXCR3 (0.57) SMN1; SMN2ALDH1A1NPSR1MAPK1CXCR3
SCHEMBL7144891 0.73 CXCR3 (0.62) PDE10ACXCR3
SCHEMBL450061 0.73 CXCR3 (0.54) SMN1; SMN2ALDH1A1KMT2AMEN1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083190-A1 INSECT ODORANT RECEPTOR ANTAGONISTS THE ROCKEFELLER UNIVERSITY (US) 2012-06-21 WO disclosed