SCHEMBL9970820

SCHEMBL9970820

O=C(NC1CCCC(Nc2nc(-c3n[nH]c4ncc(F)cc34)c(F)cc2F)C1)c1ccsc1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.37
CDK7 P50613 1/20 0.36
BTK Q06187 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15401564 1.00 GRM5 (0.37) GRM5CDK7BTK
SCHEMBL9977728 0.91 GSK3A (0.39) GRM5
SCHEMBL15399800 0.91 GSK3A (0.39) GRM5
SCHEMBL16199061 0.91 GSK3A (0.39) GRM5
SCHEMBL9967246 0.88 CDK7 (0.43) CDK7
SCHEMBL15401369 0.87 CDK7 (0.38) GRM5CDK7
SCHEMBL9970812 0.87 CDK7 (0.38) GRM5CDK7
SCHEMBL9970823 0.81 BTK (0.34) GRM5CDK7BTK
SCHEMBL15401427 0.80 GSK3A (0.39)
SCHEMBL15400659 0.80 GSK3A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083121-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-21 WO disclosed