SCHEMBL9972174

SCHEMBL9972174

CSc1nc2sc3c(c2c(=O)[nH]1)CCC3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
HPGD P15428 5/20 1.00
SMN1; SMN2 Q16637 2/20 0.70
MAPT P10636 3/20 0.68
LMNA P02545 1/20 0.65
RAB9A P51151 1/20 0.65
HIF1A Q16665 2/20 0.63
CYP1A2 P05177 1/20 0.63
CDKN1A P38936 1/20 0.62
PARP1 P09874 2/20 0.59
KDM4E B2RXH2 2/20 0.58
MEN1 O00255 1/20 0.58
GAA P10253 1/20 0.58
HTT P42858 1/20 0.58
KMT2A Q03164 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
ADORA3 P0DMS8 1/20 0.57
BRD4 O60885 3/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7992628 0.80 ALDH1A1 (0.67) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL21637701 0.78 KDM4E (0.70) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL1368527 0.78 HIF1A (1.00) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL3924721 0.78 SMN1; SMN2 (0.73) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL541201 0.78 LMNA (0.76) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL12281819 0.77 SMN1; SMN2 (0.72) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL1368915 0.75 ALDH1A1 (0.71) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL8190292 0.74 ALDH1A1 (0.65) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL13155648 0.74 ALDH1A1 (0.65) ALDH1A1HPGDSMN1; SMN2MAPTHIF1A
SCHEMBL8198190 0.73 ALDH1A1 (0.63) ALDH1A1HPGDSMN1; SMN2MAPTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8202861-B2 Drugs for various disorders VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-19 US disclosed
US-8202861-B2 Drugs for various disorders VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-19 US disclosed